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Search Results for " anti-proliferative activity "

20

Compounds

Cat No. Product Name Synonyms Targets
T1687 Doxycycline Vibramycin,Doxiciclina,Doxytetracycline,Doxycyclinum MMP , ribosome , Antibacterial , Antibiotic , Parasite
Doxycycline (Doxiciclina) belongs to the tetracycline class of antibiotics and is a broad-spectrum metalloproteinase (MMP) inhibitor with oral activity. Doxycycline has antibacterial activity and antitumor activity.
T1687L Doxycycline (hyclate) Doxycycline hydrochloride hemiethanolate hemihydrate,WC2031,Doxycycline hyclate MMP , ribosome , Antibacterial , Antibiotic
Doxycycline hyclate (WC2031) belongs to the tetracycline class of antibiotics and is a broad-spectrum metalloproteinase (MMP) inhibitor with oral activity. Doxycycline hyclate has antibacterial activity and antitumor act...
T12477 Uzansertib phosphate INCB053914 phosphate Pim
Uzansertib phosphate (INCB053914 phosphate) is an orally active, ATP-competitive inhibitor of pan-PIM kinase(PIM1, PIM2, PIM3 with IC50s of 0.24 nM, 30 nM, 0.12 nM , respectively).
T5858 Sertindole Lu 23-174 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Autophagy
Sertindole (Lu 23-174) is an atypical antipsychotic that binds to dopamine D2 receptors and the serotonin (5-HT) receptor subtypes 5-HT1D, 5-HT2A, and 5-HT2C (Kds = 2.7, 20, 0.14, and 6 nM, respectively)
T5135 Flupentixol dihydrochloride Fupentixol Dihydrochloride,Flupenthixol dihydrochloride,(E/Z)-Flupentixol Dihydrochloride Dopamine Receptor
Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.
T1140 Doxycycline hydrochloride Doxylin,Vibramycin,Hyclate MMP , Antibacterial , Antibiotic
Doxycycline hydrochloride (Hyclate) is a synthetic tetracycline derivative with similar antimicrobial activity.
TQ0134 Podocarpusflavone A Topoisomerase
Podocarpusflavone A is a DNA topoisomerase I inhibitor. It has moderated anti-proliferative activity induce cell apoptosis in MCF-7.
T60225 Biguanidinium-porphyrin Others
Biguanidinium-porphyrin is a phototoxic agent with anti-proliferative activity.
T5S0803 Columbamine Columbamin,Dehydroisocorypalmine Others
Columbamine (Columbamin) shows strong activity with IC5 48.1 μM.Columbamine exerts anti-proliferative and anti-vasculogenic effects on metastatic human osteosarcoma U2OS cells with low toxicity.
T9582 CLEFMA NF-κB
CLEFMA has anti-proliferative activity. CLEFMA inhibits tumor growth associated with NF-κB-regulated anti-inflammatory and anti-metastatic effects.
T10111 3-Deazaadenosine hydrochloride Others , HIV Protease
3-Deazaadenosine hydrochloride is an inhibitor of S-adenosylhomocysteine hydrolase (Ki: 3.9 µM). It has anti-inflammatory, anti-proliferative, and anti-HIV activity.
TMS0943 Platicodigenin Platycodigenin Others
Platicodigenin (Platycodigenin) isolated from platycodon grandiflorum, has in vitro anti-proliferative activity against the HSC-T6 cell line.
T60852 Anticancer agent 46
Anticancer agent 46 is a potent anti-cancer agent, showing anti-proliferative activity in cellular assays, with an IC50 of 0.986 μM against MGC803 cells.
T6S1683 Demethoxycurcumin Curcumin II,Desmethoxycurcumin,Monodemethoxycurcumin Apoptosis , Antioxidant , Antibacterial , Autophagy
1. Demethoxycurcumin (Desmethoxycurcumin) has antioxidant activity. 2. Demethoxycurcumin has anti-inflammatory activity. 3. Demethoxycurcumin has anti-proliferative activity. 4. Demethoxycurcumin has anti-acanthamoebic e...
TQ0318 Filanesib ARRY-520,ARRY 520 KSP
Filanesib (ARRY 520) is a selective inhibitor of kinesin spindle protein (KSP, IC50 = 6 nM) with potent anti-proliferative activity.
T10882 CPUY074020 Histone Methyltransferase
CPUY074020 is a potent and orally bioavailable inhibitor of histone methyltransferase G9a (IC50: 2.18 μM) with anti-proliferative activity.
T77728 Tubulin polymerization-IN-55 Microtubule Associated
Tubulin polymerization-IN-55 is a potent Tubulin Polymerization inhibitor with potential anti-angiogenic and anti-tumour activity, showing anti-proliferative effects against A549, K562, HepG2, MDA-MB-231 and HFL-1.
T60753 L82 DNA
L82 is a DNA ligase 1 (DNA Lig1) inhibitor (hLig1 IC50=12 μM) that is selective and non-competitive.L82 expresses anti-proliferative activity against breast cancer cells.
T3796 Betulinaldehyde Betulinic aldehyde,Betulinal,Betunal Apoptosis , Antibacterial
Betulinaldehyde (Betunal) has the inhibition of Saccharomyces sp and alpha-glucosidase. Betulinaldehyde induces apoptosis in mouse B16 2F2 cells. Betulinaldehyde has anti-proliferative activity against mouse +SA mammary ...
TQ0318L ARRY 520 hydrochloride KSP
ARRY 520 hydrochloride is a kinesin spindle protein (KSP) inhibitor.ARRY 520 hydrochloride induces cell death by apoptosis and has potent anti-proliferative activity.

Compounds

Doxycycline
T1687
Synonym: Vibramycin,Doxiciclina,Doxytetracycline,Doxycyclinum
Target: MMP, ribosome, Antibacterial, Antibiotic, Parasite
Doxycycline (hyclate)
T1687L
Synonym: Doxycycline hydrochloride hemiethanolate hemihydrate,WC2031,Doxycycline hyclate
Target: MMP, ribosome, Antibacterial, Antibiotic
Uzansertib phosphate
T12477
Synonym: INCB053914 phosphate
Target: Pim
Sertindole
T5858
Synonym: Lu 23-174
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Autophagy
Flupentixol dihydrochloride
T5135
Synonym: Fupentixol Dihydrochloride,Flupenthixol dihydrochloride,(E/Z)-Flupentixol Dihydrochloride
Target: Dopamine Receptor
Doxycycline hydrochloride
T1140
Synonym: Doxylin,Vibramycin,Hyclate
Target: MMP, Antibacterial, Antibiotic
Podocarpusflavone A
TQ0134
Synonym:
Target: Topoisomerase
Biguanidinium-porphyrin
T60225
Synonym:
Target: Others
Columbamine
T5S0803
Synonym: Columbamin,Dehydroisocorypalmine
Target: Others
CLEFMA
T9582
Synonym:
Target: NF-κB
3-Deazaadenosine hydrochloride
T10111
Synonym:
Target: Others, HIV Protease
Platicodigenin
TMS0943
Synonym: Platycodigenin
Target: Others
Anticancer agent 46
T60852
Synonym:
Target:
Demethoxycurcumin
T6S1683
Synonym: Curcumin II,Desmethoxycurcumin,Monodemethoxycurcumin
Target: Apoptosis, Antioxidant, Antibacterial, Autophagy
Filanesib
TQ0318
Synonym: ARRY-520,ARRY 520
Target: KSP
CPUY074020
T10882
Synonym:
Target: Histone Methyltransferase
Tubulin polymerization-IN-55
T77728
Synonym:
Target: Microtubule Associated
L82
T60753
Synonym:
Target: DNA
Betulinaldehyde
T3796
Synonym: Betulinic aldehyde,Betulinal,Betunal
Target: Apoptosis, Antibacterial
ARRY 520 hydrochloride
TQ0318L
Synonym:
Target: KSP
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TargetMol